Lobeline hydrochloride
CAS No. 134-63-4
Lobeline hydrochloride ( Lobeline hydrochloride )
Catalog No. M11393 CAS No. 134-63-4
Lobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes.
Purity : >98%(HPLC)
Size | Price / USD | Stock | Quantity |
50MG | 41 | In Stock |
|
100MG | 74 | In Stock |
|
200MG | 87 | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameLobeline hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionLobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes.
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DescriptionLobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes.
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SynonymsLobeline hydrochloride
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PathwayEndocrinology/Hormones
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TargetAChR
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RecptornAChR; Nicotinic Receptor
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Research AreaNeurological Disease
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Indication——
Chemical Information
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CAS Number134-63-4
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Formula Weight273.92
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Molecular FormulaC22H27NO2·HCl
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Purity>98%(HPLC)
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SolubilityWater: 1g/40mL
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SMILESCN1[C@@H](CC(C2=CC=CC=C2)=O)CCC[C@H]1C[C@H](O)C3=CC=CC=C3.[H]Cl
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Chemical Name2-[(2R,6S)-6-[(2S)-2-Hydroxy-2-phenylethyl]-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Dichlorisone Acetate
It belongs to organophosphate compounds, used as a kind of common environmental health insecticide.
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PHA 568487
The quinuclidine PHA 568487 is an agonist of the alpha 7 nicotinic acetylcholine receptor that was designed to mitigate the bioactivation associated with the core scaffold and subsequently remove associated liabilities with in vivo tolerability.
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Catestatin
Non-competitive nicotinic cholinergic antagonist; selectively inhibits nicotinic-stimulated catecholamine secretion from chromaffin cells and noradrenergic neurons (IC50 ~ 200 nM). Blocks nicotinic-induced cationic signaling (IC50 ~ 200 - 250 nM) and inhibits nicotinic-agonist induced desensitization of catecholamine release. Also stimulates mast cell release of histamine via a separate mechanism.